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RS 127445
CAS No. 199864-86-3
RS 127445 ( MT 500 )
Catalog No. M20836 CAS No. 199864-86-3
RS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 42 | In Stock |
|
| 10MG | 69 | In Stock |
|
| 25MG | 131 | In Stock |
|
| 50MG | 236 | In Stock |
|
| 100MG | 356 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRS 127445
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NoteResearch use only not for human use.
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Brief DescriptionRS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
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DescriptionRS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
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SynonymsMT 500
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT2B
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Research Area——
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Indication——
Chemical Information
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CAS Number199864-86-3
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Formula Weight317.79
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Molecular FormulaC17H17ClFN3
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Purity>98% (HPLC)
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SolubilityDMSO:31 mg/mL (97.55 mM)
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SMILESCC(C)c1cc(-c2ccc(F)c3ccccc23)nc(N)n1.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Bonhaus D W Flippin L A Greenhouse R J et al. RS-127445: a selective high affinity orally bioavailable 5-HT2B receptor antagonist[J]. 1999 127(5):1075-1082.
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