RS 127445
CAS No. 199864-86-3
RS 127445 ( MT 500 )
Catalog No. M20836 CAS No. 199864-86-3
RS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 42 | In Stock |
|
10MG | 69 | In Stock |
|
25MG | 131 | In Stock |
|
50MG | 236 | In Stock |
|
100MG | 356 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
-
Product NameRS 127445
-
NoteResearch use only not for human use.
-
Brief DescriptionRS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
-
DescriptionRS 127445 is a selective high affinity orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).
-
SynonymsMT 500
-
PathwayEndocrinology/Hormones
-
Target5-HT Receptor
-
Recptor5-HT2B
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number199864-86-3
-
Formula Weight317.79
-
Molecular FormulaC17H17ClFN3
-
Purity>98% (HPLC)
-
SolubilityDMSO:31 mg/mL (97.55 mM)
-
SMILESCC(C)c1cc(-c2ccc(F)c3ccccc23)nc(N)n1.Cl
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Bonhaus D W Flippin L A Greenhouse R J et al. RS-127445: a selective high affinity orally bioavailable 5-HT2B receptor antagonist[J]. 1999 127(5):1075-1082.
molnova catalog
related products
-
Espindolol
Espindolol is a novel non-selective β blocker with central 5-HT1a and partial β2 receptor agonist effects.
-
Dalasetron Mesylate ...
Dolasetron(MDL-73147) is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy.
-
Iloperidone hydrochl...
An atypical antipsychotic that exhibits high affinity to serotonin 5HT2A (Ki =5.6 nM), dopamine D2 (Ki=6.3 nM) and D3 (Ki=7.1 nM) and noradrenaline α1 receptors (Ki=0.36 nM).